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Exploring the structural and functional requirements of Phyto-compounds and their synthetic scaffolds as anticancer agents: Medicinal chemistry perspective - ScienceDirect
Exploring the structural and functional requirements of Phyto-compounds and their synthetic scaffolds as anticancer agents: Medicinal chemistry perspective - ScienceDirect

Structural Evolution and Translational Potential for Agonists and Antagonists of Endosomal Toll-like Receptors | Journal of Medicinal Chemistry
Structural Evolution and Translational Potential for Agonists and Antagonists of Endosomal Toll-like Receptors | Journal of Medicinal Chemistry

Protein‐Templated Fragment Ligations—From Molecular Recognition to Drug Discovery - Jaegle - 2017 - Angewandte Chemie International Edition - Wiley Online Library
Protein‐Templated Fragment Ligations—From Molecular Recognition to Drug Discovery - Jaegle - 2017 - Angewandte Chemie International Edition - Wiley Online Library

Morpholine as ubiquitous pharmacophore in medicinal chemistry: Deep insight into the structure-activity relationship (SAR) - ScienceDirect
Morpholine as ubiquitous pharmacophore in medicinal chemistry: Deep insight into the structure-activity relationship (SAR) - ScienceDirect

Molecules | Free Full-Text | Synthesis and Evaluation of NF-κB Inhibitory Activity of Mollugin Derivatives
Molecules | Free Full-Text | Synthesis and Evaluation of NF-κB Inhibitory Activity of Mollugin Derivatives

Synthetic Approaches to the New Drugs Approved During 2017 | Journal of Medicinal Chemistry
Synthetic Approaches to the New Drugs Approved During 2017 | Journal of Medicinal Chemistry

Bioactive Aurones, Indanones, and Other Hemiindigoid Scaffolds: Medicinal Chemistry and Photopharmacology Perspectives | Journal of Medicinal Chemistry
Bioactive Aurones, Indanones, and Other Hemiindigoid Scaffolds: Medicinal Chemistry and Photopharmacology Perspectives | Journal of Medicinal Chemistry

Bioorganic & Medicinal Chemistry Letters | Vol 27, Issue 3, Pages 361-700 (1 February 2017) | ScienceDirect.com by Elsevier
Bioorganic & Medicinal Chemistry Letters | Vol 27, Issue 3, Pages 361-700 (1 February 2017) | ScienceDirect.com by Elsevier

Nonconjugated Hydrocarbons as Rigid‐Linear Motifs: Isosteres for Material Sciences and Bioorganic and Medicinal Chemistry - Locke - 2019 - Chemistry – A European Journal - Wiley Online Library
Nonconjugated Hydrocarbons as Rigid‐Linear Motifs: Isosteres for Material Sciences and Bioorganic and Medicinal Chemistry - Locke - 2019 - Chemistry – A European Journal - Wiley Online Library

Targeting Stimulator of Interferon Genes (STING): A Medicinal Chemistry Perspective | Journal of Medicinal Chemistry
Targeting Stimulator of Interferon Genes (STING): A Medicinal Chemistry Perspective | Journal of Medicinal Chemistry

Molecules | Free Full-Text | Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–5
Molecules | Free Full-Text | Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–5

Design of Novel 3-Pyrimidinylazaindole CDK2/9 Inhibitors with Potent In Vitro and In Vivo Antitumor Efficacy in a Triple-Negative Breast Cancer Model | Journal of Medicinal Chemistry
Design of Novel 3-Pyrimidinylazaindole CDK2/9 Inhibitors with Potent In Vitro and In Vivo Antitumor Efficacy in a Triple-Negative Breast Cancer Model | Journal of Medicinal Chemistry

Recent Advances in the Medicinal Chemistry of Farnesoid X Receptor | Journal of Medicinal Chemistry
Recent Advances in the Medicinal Chemistry of Farnesoid X Receptor | Journal of Medicinal Chemistry

Discovery and Optimization of Boronic Acid Based Inhibitors of Autotaxin | Journal of Medicinal Chemistry
Discovery and Optimization of Boronic Acid Based Inhibitors of Autotaxin | Journal of Medicinal Chemistry

Discovery of Novel Small-Molecule Inhibitors of NF-κB Signaling with Antiinflammatory and Anticancer Properties | Journal of Medicinal Chemistry
Discovery of Novel Small-Molecule Inhibitors of NF-κB Signaling with Antiinflammatory and Anticancer Properties | Journal of Medicinal Chemistry

Molecules | Free Full-Text | Pharmacotherapeutics Applications and Chemistry of Chalcone Derivatives
Molecules | Free Full-Text | Pharmacotherapeutics Applications and Chemistry of Chalcone Derivatives

Medicinal chemistry of indole derivatives: Current to future therapeutic prospectives - ScienceDirect
Medicinal chemistry of indole derivatives: Current to future therapeutic prospectives - ScienceDirect

Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration | Journal of Medicinal Chemistry
Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration | Journal of Medicinal Chemistry

Molecules | Free Full-Text | Boron Chemicals in Drug Discovery and Development: Synthesis and Medicinal Perspective
Molecules | Free Full-Text | Boron Chemicals in Drug Discovery and Development: Synthesis and Medicinal Perspective

Structure-Based Discovery of New Antagonist and Biased Agonist Chemotypes for the Kappa Opioid Receptor | Journal of Medicinal Chemistry
Structure-Based Discovery of New Antagonist and Biased Agonist Chemotypes for the Kappa Opioid Receptor | Journal of Medicinal Chemistry

Molecules | Free Full-Text | Efforts in Bioprospecting Research: A Survey of Novel Anticancer Phytochemicals Reported in the Last Decade
Molecules | Free Full-Text | Efforts in Bioprospecting Research: A Survey of Novel Anticancer Phytochemicals Reported in the Last Decade

Molecules | Free Full-Text | Chlojaponilactone B Attenuates Lipopolysaccharide-Induced Inflammatory Responses by Suppressing TLR4-Mediated ROS Generation and NF-κB Signaling Pathway
Molecules | Free Full-Text | Chlojaponilactone B Attenuates Lipopolysaccharide-Induced Inflammatory Responses by Suppressing TLR4-Mediated ROS Generation and NF-κB Signaling Pathway

Structure-Based Design of Tricyclic NF-κB Inducing Kinase (NIK) Inhibitors That Have High Selectivity over Phosphoinositide-3-kinase (PI3K) | Journal of Medicinal Chemistry
Structure-Based Design of Tricyclic NF-κB Inducing Kinase (NIK) Inhibitors That Have High Selectivity over Phosphoinositide-3-kinase (PI3K) | Journal of Medicinal Chemistry

Drug Discovery: Covalent Bonds Between Small Molecules & Proteins
Drug Discovery: Covalent Bonds Between Small Molecules & Proteins

Molecules | Free Full-Text | Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–7
Molecules | Free Full-Text | Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–7

PDF) Synthesis and antibacterial evaluation of macrocyclic diarylheptanoid derivatives | Aman Singh - Academia.edu
PDF) Synthesis and antibacterial evaluation of macrocyclic diarylheptanoid derivatives | Aman Singh - Academia.edu

Molecules | Free Full-Text | Anti-Cancer Potential of Synthetic Oleanolic Acid Derivatives and Their Conjugates with NSAIDs
Molecules | Free Full-Text | Anti-Cancer Potential of Synthetic Oleanolic Acid Derivatives and Their Conjugates with NSAIDs

Scaffold Diversity Inspired by the Natural Product Evodiamine: Discovery of Highly Potent and Multitargeting Antitumor Agents | Journal of Medicinal Chemistry
Scaffold Diversity Inspired by the Natural Product Evodiamine: Discovery of Highly Potent and Multitargeting Antitumor Agents | Journal of Medicinal Chemistry

Molecules | Free Full-Text | 2-Phenethylamines in Medicinal Chemistry: A Review
Molecules | Free Full-Text | 2-Phenethylamines in Medicinal Chemistry: A Review

Targeting the Receptor for Advanced Glycation Endproducts (RAGE): A Medicinal Chemistry Perspective | Journal of Medicinal Chemistry
Targeting the Receptor for Advanced Glycation Endproducts (RAGE): A Medicinal Chemistry Perspective | Journal of Medicinal Chemistry

4‐(Di‐/Trifluoromethyl)‐2‐heterabicyclo[2.1.1]hexanes: Advanced Fluorinated Phenyl Isosteres and Proline analogues - Homon - 2021 - European Journal of Organic Chemistry - Wiley Online Library
4‐(Di‐/Trifluoromethyl)‐2‐heterabicyclo[2.1.1]hexanes: Advanced Fluorinated Phenyl Isosteres and Proline analogues - Homon - 2021 - European Journal of Organic Chemistry - Wiley Online Library

Bioorganic & Medicinal Chemistry | From controlling chemical bonding to deciphering and manipulating biological processes | ScienceDirect.com by Elsevier
Bioorganic & Medicinal Chemistry | From controlling chemical bonding to deciphering and manipulating biological processes | ScienceDirect.com by Elsevier

The Cravatt Lab
The Cravatt Lab

Bioorganic & Medicinal Chemistry | Vol 10, Issue 12, Pages 3695-4194 (December 2002) | ScienceDirect.com by Elsevier
Bioorganic & Medicinal Chemistry | Vol 10, Issue 12, Pages 3695-4194 (December 2002) | ScienceDirect.com by Elsevier

Synthesis and Biological Evaluation of Derivatives of Indoline as Highly Potent Antioxidant and Anti-inflammatory Agents | Journal of Medicinal Chemistry
Synthesis and Biological Evaluation of Derivatives of Indoline as Highly Potent Antioxidant and Anti-inflammatory Agents | Journal of Medicinal Chemistry

Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases | Journal of Medicinal Chemistry
Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases | Journal of Medicinal Chemistry

Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design | Journal of Medicinal Chemistry
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design | Journal of Medicinal Chemistry

The Cravatt Lab
The Cravatt Lab

Molecules | Free Full-Text | Chemistry and the Potential Antiviral, Anticancer, and Anti-Inflammatory Activities of Cardiotonic Steroids Derived from Toads
Molecules | Free Full-Text | Chemistry and the Potential Antiviral, Anticancer, and Anti-Inflammatory Activities of Cardiotonic Steroids Derived from Toads

Are We Opening the Door to a New Era of Medicinal Chemistry or Being Collapsed to a Chemical Singularity? | Journal of Medicinal Chemistry
Are We Opening the Door to a New Era of Medicinal Chemistry or Being Collapsed to a Chemical Singularity? | Journal of Medicinal Chemistry